產品標題 |
俗名 |
產品學名 |
英文品名 |
結構式 |
CAS NO |
可制成原料藥 |
艾氟康唑中間體 Efinaconazole ITS-1 |
艾氟康唑中間體 Efinaconazole ITS-1 |
1.1 - (((2R,3S)-2-(2,4-二氟苯基)-3-甲基環氧乙烷-2-基)甲基)-1H-1,2,4-三唑 |
1. 1-(((2R, 3S)-2-(2,4-difluorophenyl)-3-Methyloxiran-2-yl) Methyl)-1H-1,2,4-triazole |
 |
127000-90-2 |
艾氟康唑 Efinaconazole |
艾莎康唑中間體-5 Isavuconazole ITS-5 |
艾莎康唑中間體-5 Isavuconazole ITS-5 |
1-[[(2R,3S)-2-(2,5-二氟苯基)-3-甲基環氧乙烷基]甲基]-1H-1,2,4-三唑 |
1-(((2R,3S)-2-(2,5-difluorophenyl)-3-Methyloxiran-2-yl)Methyl)-1H-1,2,4-triazole |
 |
241479-73-2 |
艾莎康唑 Isavuconazole |
艾莎康唑中間體-4 Isavuconazole ITS-4 |
艾莎康唑中間體-4 Isavuconazole ITS-4 |
(2R)-2',5'-二氟-2-(3,4,5,6-四氫-2H-吡喃-2-基氧基)-苯乙酮 |
(2R)-2',5'-difluoro-2-(3,4,5,6-tetrahydro-2H-pyran-2-yloxy)-propiophenone |
 |
241479-69-6 |
艾莎康唑 Isavuconazole |
艾莎康唑中間體-3 Isavuconazole ITS-3 |
艾莎康唑中間體-3 Isavuconazole ITS-3 |
(2S)-1-(4-嗎啉基)-2-[(四氫-2H-吡喃-2-基)氧基]-1-丙酮 |
(2S)-1-Morpholin-4-yl-2-(tetrahydro-pyran-2-yloxy)-propan-1-one |
 |
135206-86-9 |
艾莎康唑 Isavuconazole |
艾莎康唑中間體-2 Isavuconazole ITS-2 |
艾莎康唑中間體-2 Isavuconazole ITS-2 |
\ |
\ |
 |
1110002-01-0 |
艾莎康唑 Isavuconazole |
艾莎康唑中間體-1 Isavuconazole ITS-1 |
艾莎康唑中間體-1 Isavuconazole ITS-1 |
(2R,3R)-3-(2,5-二氟苯基)-3-羥基-2-甲基-4-(1H-(1,2,4)-三氮唑-1-基)硫代丁酰胺硫酸鹽一水合物 |
(2R,3R)-3-(2,5-Difluorophenyl)-3-hydroxy-2-Methyl-4-(1H-1,2,4-triazol-1-yl)thiobutyraMide |
 |
368421-58-3 |
艾莎康唑 Isavuconazole |
氨磺必利中間體 Amisulpride ITS |
氨磺必利中間體 Amisulpride ITS |
2-甲氧基-4-氨基-5-乙磺酰苯甲酸 |
4-Amino-5-ethylsulfonyl-2-methoxybenzoic acid |
 |
71675-87-1 |
氨磺必利 Amisulpride |
瑞巴派特中間體-2 Rebamipide ITS-2 |
瑞巴派特中間體-2 Rebamipide ITS-2 |
\ |
Rebamipide sodium |
 |
\ |
瑞巴派特 Rebamipide |
瑞巴派特中間體-1 Rebamipide ITS-1 |
瑞巴派特中間體-1 Rebamipide ITS-1 |
2-氨基-3-(2-氧代-1,2-二氫喹啉-4-基)丙酸二鹽酸鹽二水合物 |
4-Quinolinepropanoic acid, α-amino-1,2-dihydro-2-oxo-, dihydrochloride, dihydrate |
 |
914769-50-9 |
瑞巴派特 Rebamipide |
托伐普坦中間體 Tolvaptan ITS |
托伐普坦中間體 Tolvaptan ITS |
7-氯-1,2,3,4-四氫苯并[B]氮雜卓-5-酮 |
7-CHLORO-1,2,3,4-TETRAHYDRO-BENZO[B]AZEPIN-5-ONE |
 |
160129-45-3 |
托伐普坦 Tolvaptan |
立他司特中間體-3 Lifitegrast ITS-3 |
立他司特中間體-3 Lifitegrast ITS-3 |
苯并呋喃-6-羧酸 |
6-Benzofurancarboxylic acid |
 |
77095-51-3 |
立他司特 Lifitegrast |
立他司特中間體-2 Lifitegrast ITS-2 |
立他司特中間體-2 Lifitegrast ITS-2 |
\ |
\ |
 |
1194550-59-8 (R=Bn) 851785-21-2 (R=Me) 1270093-99-6 (R=H) |
立他司特 Lifitegrast |
立他司特中間體-1 Lifitegrast ITS-1 |
立他司特中間體-1 Lifitegrast ITS-1 |
\ |
\ |
 |
851784-82-2 (R1=H, R2=Boc) 851784-80-0(R1=Me, R2=Boc) 1289646-93-0 (R1=H, R2=H) 851784-90-2 (R1=Me, R2=H) |
立他司特 Lifitegrast |
帕博西尼 Palbociclib base |
帕博西尼 Palbociclib base |
帕博西尼 |
palbociclib |
 |
571190-30-2 |
帕博西林鹽酸鹽Palbociclib Hydrochloride |
帕博西林中間體-3 Palbociclib ITS-3 |
帕博西林中間體-3 Palbociclib ITS-3 |
\ |
\ |
 |
866084-31-3(R=n-Butyl) 571189-10-1(R=Ethyl) |
帕博西林鹽酸鹽Palbociclib Hydrochloride |
帕博西林中間體-2 Palbociclib ITS-2 |
帕博西林中間體-2 Palbociclib ITS-2 |
4-(6-氨基吡啶-3-基)哌嗪-1-羧酸叔丁酯 |
tert-Butyl 4-(6-aminopyridin-3-yl)piperazine-1-carboxylate |
 |
571188-59-5 |
帕博西林鹽酸鹽Palbociclib Hydrochloride |
帕博西林中間體-1 Palbociclib ITS-1 |
帕博西林中間體-1 Palbociclib ITS-1 |
6-溴-2-氯-8-環戊基-5-甲基-吡啶并[2,3-D]嘧啶-7(8H)-酮 |
6-broMo-2-chloro-8-cyclopentyl-5-Methylpyrido[2,3-d]pyriMidin-7(8H)-one |
 |
1016636-76-2 |
帕博西林鹽酸鹽Palbociclib Hydrochloride |
克立硼羅中間體-3 Crisaborole ITS-3 |
克立硼羅中間體-3 Crisaborole ITS-3 |
4-[4-溴-3-(羥基甲基)苯氧基]苯甲腈 |
4-(4-broMo-3-(hydroxyMethyl)phenoxy)benzonitrile |
 |
906673-45-8 |
克立硼羅 Crisaborole |
克立硼羅中間體-2 Crisaborole ITS-2 |
克立硼羅中間體-2 Crisaborole ITS-2 |
4-(4-溴-3-甲?;窖趸?苯甲腈 |
4-(4-Bromo-3-formyl-phenoxy)-benzonitrile |
 |
906673-54-9 |
克立硼羅 Crisaborole |
克立硼羅中間體-1 Crisaborole ITS-1 |
克立硼羅中間體-1 Crisaborole ITS-1 |
2-溴-5-羥基苯甲醛 |
2-BROMO-5-HYDROXYBENZALDEHYDE |
 |
2973-80-0 |
克立硼羅 Crisaborole |
卡培他濱中間體Cap-6 Capecitabine ITS Cap-6 |
卡培他濱中間體Cap-6 Capecitabine ITS Cap-6 |
5'-脫氧-5-氟-N-[(戊氧基)羰基]胞苷 2',3'-二乙酸酯 |
5`-deoxy-5-fluore-N-[(pentoyloxy)carbonyl]cytidine 2`,3`-diacetate |
 |
162204-20-8 |
卡培他濱 Capecitabine |
卡培他濱中間體Cap-5 Capecitabine ITS Cap-5 |
卡培他濱中間體Cap-5 Capecitabine ITS Cap-5 |
2',3'-二-O-乙?;?5'-脫氧-5-氟-D-胞啶 |
2',3'-Di-O-acetyl-5'-deoxy-5-fluoro-D-cytidine |
 |
161599-46-8 |
卡培他濱 Capecitabine |
卡培他濱中間體Cap-4 Capecitabine ITS Cap-4 |
卡培他濱中間體Cap-4 Capecitabine ITS Cap-4 |
1,2,3-三乙酰氧基-5-脫氧-D-核糖 |
1,2,3-Triacetyl-5-deoxy-D-ribose |
 |
62211-93-2 |
卡培他濱 Capecitabine |
吉西他濱中間體-T9 Gemcitabine ITS-T9 |
吉西他濱中間體-T9 Gemcitabine ITS-T9 |
2',2'-二氟-2'-脫氧胞嘧啶核苷-3',5'-二苯甲酸酯 |
2',2'-Difluoro-2'-deoxycytidine-3',5'-dibenzoate |
 |
134790-39-9 |
吉西他濱 Gemcitabine |
吉西他濱中間體-T8 Gemcitabine ITS-T8 |
吉西他濱中間體-T8 Gemcitabine ITS-T8 |
2-脫氧-2,2-二氟-D-赤式-五呋喃糖-3,5-二苯甲酯-1-甲磺酸酯 |
2-deoxy-2,2-difluoro-d-erythro-pentofuranose-3,5-dibenzoate-1-methanesulfonate |
 |
122111-11-9 |
吉西他濱 Gemcitabine |